Protein Details: Neuronal acetylcholine receptor subunit alpha-4

Protein ID

ICDB_Pro_0857

Protein Name

Neuronal acetylcholine receptor subunit alpha-4

Gene Name

CHRNA4

Organism

Mustela putorius furo (European domestic ferret) (Mustela furo)

Length

627 amino acids

AlphaFoldDB

AF-Q19AE6-F1-model_v4.pdb

Function

After binding acetylcholine; the AChR responds by an extensive change in conformation that affects all subunits and leads to opening of an ion-conducting channel across the plasma membrane.

Sequence

MELGGPGAPPPPLLPPLLLLLGAGFLPASSPVETRAHAEERLLKTLFSGYNKWSRPVANISDVVLVHFGLSIAQLIDVDEKNQMMTTNVWVKQEWYDYKLRWDPADYENVTSIRIPSELIWRPDIVLYNNADGDFAITHLTKAHLFHDGRVQWTPPAIYKSSCSIDVTFFPFDQQNCTMKFGSWTYDKAKIDLVSMQSHVDQLGLWESGEWVIVDAAGTYNTRKYECCAEVYPDITYAFVIRRLPLFYTINLIVPCLLISCLTVLVFYLPSDCGEKVTLCISVLLSLTVFLLLITEIIPSTSLVIPLIGEYLLFTMVFVTLSIVITVFVLNVHHRSPRTHTMPAWVRRVFLDVVPRLLLMKRPSVVKDNCRRLIESMHKVASAPGFWPEPEGEPGVVSGERSRGPSRSASFRGPRDEPAEPQPACASPSDRVPAPQPSEGDPGSPCPLPDSCRPPPSTRAPGLTEARSLSFQHVSSAAERVEGGVRCRSWSIQGCAPQDEAASVAGGPVTSSPAFPKASAAELLPPDQPSPCRCRCRKEPSPNAVRKACGTRVPARHLPLSPALARAVEGVQYIADHLKAEDTDFSVKEDWKYVAMVIDRIFLWVFVIVCLLGTAGLFLPPWLAGMI

PDB Structures

Ligand Binding

1. DICL_CP

2. DICL_Pep

Binding Site

Disease

Location

DOI ID

10.1124/mol.51.2.320

RefSeq

NP_990695.1

Feature